Academic Journal

Four new cytotoxic triterpenoids from Euphorbia fischeriana.

Λεπτομέρειες βιβλιογραφικής εγγραφής
Τίτλος: Four new cytotoxic triterpenoids from Euphorbia fischeriana.
Συγγραφείς: He YB; Yunnan Key Laboratory of Modern Separation Analysis and Substance Transformation, Faculty of Chemistry and Chemical Engineering, Yunnan Normal University, Kunming, China., Ma YN; Kunming Municipal Hospital of Traditional Chinese Medicine, Yunnan University of Traditional Chinese Medicine, Kunming, China., Huang YP; Yunnan Key Laboratory of Modern Separation Analysis and Substance Transformation, Faculty of Chemistry and Chemical Engineering, Yunnan Normal University, Kunming, China., Li WN; Yunnan Key Laboratory of Modern Separation Analysis and Substance Transformation, Faculty of Chemistry and Chemical Engineering, Yunnan Normal University, Kunming, China., Shi TX; Yunnan Key Laboratory of Modern Separation Analysis and Substance Transformation, Faculty of Chemistry and Chemical Engineering, Yunnan Normal University, Kunming, China., Yang J; State Key Laboratory of Phytochemistry and Plant Resources in West China, Kunming Institute of Botany, Chinese Academy of Sciences, Kunming, China., Zhao Y; Yunnan Key Laboratory of Modern Separation Analysis and Substance Transformation, Faculty of Chemistry and Chemical Engineering, Yunnan Normal University, Kunming, China.
Πηγή: Natural product research [Nat Prod Res] 2026 Jul; Vol. 40 (14), pp. 4136-4146. Date of Electronic Publication: 2025 May 16.
Τύπος έκδοσης: Journal Article
Γλώσσα: English
Στοιχεία περιοδικού: Publisher: Taylor & Francis Health Sciences Country of Publication: England NLM ID: 101167924 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1478-6427 (Electronic) Linking ISSN: 14786419 NLM ISO Abbreviation: Nat Prod Res Subsets: MEDLINE
Imprint Name(s): Original Publication: Milton Park, UK : Taylor & Francis Health Sciences, c2003-
Ιατρικοί όροι (MeSH): Euphorbia*/chemistry , Triterpenes*/chemistry , Triterpenes*/isolation & purification , Triterpenes*/pharmacology , Antineoplastic Agents, Phytogenic*/chemistry , Antineoplastic Agents, Phytogenic*/pharmacology , Antineoplastic Agents, Phytogenic*/isolation & purification, Humans ; Molecular Structure ; MCF-7 Cells ; Drug Screening Assays, Antitumor ; Inhibitory Concentration 50 ; A549 Cells
Περίληψη: Our ongoing phytochemical investigation on Euphorbia fischeriana led to isolation of four new cytotoxic triterpenoids (1-4), along with twenty three known analogues (5-27). The new structures were characterised as fiseuphanins C-F (1-4) by NMR and HRESIMS spectroscopic experiments. Among them, isolates 8-15, 17-20, 22, and 25-27 were the first examples from E. fischeriana. Compounds 2, 11, and 13 exhibited significant cytotoxic activity against MCF-7 cell line with IC50 of 0.04, 6.30, and 2.44 µM, respectively, whereas, only compounds 6, 8, 11, and 23 exhibited weak inhibitory activity against A549 with IC50 values ranging from 36.37 to 81.49 µM.
Contributed Indexing: Keywords: Euphorbia fischeriana; Euphorbiaceae; cytotoxicity; triterpenoids
Substance Nomenclature: 0 (Triterpenes)
0 (Antineoplastic Agents, Phytogenic)
Entry Date(s): Date Created: 20250516 Date Completed: 20260714 Latest Revision: 20260714
Update Code: 20260714
DOI: 10.1080/14786419.2025.2503015
PMID: 40378412
Βάση Δεδομένων: MEDLINE
Περιγραφή
ISSN:1478-6427
DOI:10.1080/14786419.2025.2503015